Mechanism of Action

Oxymetholone binds to androgen receptors in muscle tissues, stimulating protein synthesis and red blood cell production. This improves oxygen delivery to tissues, enhancing endurance and performance. It also inhibits catabolic processes that contribute to muscle breakdown.

Indications

• Treatment of anemia caused by bone marrow failure.

• Management of osteoporosis.

• Support for patients requiring significant muscle mass gain (medically supervised).

• Often used off-label in bodybuilding for performance enhancement.

Contraindications

Avoid use in individuals with:

• Hypersensitivity to Oxymetholone or any formulation components

• Severe liver disease

• Prostate cancer

• Breast cancer in men

• History of cardiovascular disorders

• Pregnant or breastfeeding women

Precautions

• Exercise caution in patients with liver dysfunction, lipid abnormalities, hypertension, or diabetes.

• Women who are pregnant or breastfeeding should not use this medication.

• Regular monitoring of liver function, blood counts, and cardiovascular status is advised.

Drug Interactions

• May interact with anticoagulants, increasing bleeding risk.

• Antidiabetic medications may be affected, altering glucose levels.

• Liver enzyme modulators may influence Oxymetholone metabolism.

• Inform healthcare providers of all medications, supplements, and substances being taken.

Dosage

• Medically supervised use depends on individual condition and response.

• Typical performance-oriented doses (not medically recommended) are 50–100 mg per day.

• Dosage adjustments should always follow medical guidance.

Storage

• Store in a dark, dry place at room temperature.

• Do not refrigerate.

• Keep out of reach of children.

Prescription Requirement

Use only under medical supervision.

Regulatory and Safety Notes

• Complies with relevant regulatory guidelines and is GMP-certified.

• Seek immediate medical attention in case of overdose.

• Report any adverse reactions to a healthcare provider.